Bojarski AJ - Search Results

1

Structure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT₃ and 5-HT₆ Receptor Antagonist with Antipsychotic and Procognitive Properties.

Zajdel P, Grychowska K, Mogilski S, Kurczab R, Satała G, Bugno R, Kos T, Gołębiowska J, Malikowska-Racia N, Nikiforuk A, Chaumont-Dubel S, Bantreil X, Pawłowski M, Martinez J, Subra G, Lamaty F, Marin P, Bojarski AJ, Popik P. Zajdel P, et al. Among authors: bojarski aj. J Med Chem. 2021 Sep 23;64(18):13279-13298. doi: 10.1021/acs.jmedchem.1c00224. Epub 2021 Sep 1. J Med Chem. 2021. PMID: 34467765 Free PMC article.

2

Structure-activity relationship studies of CNS agents--XVII. Spiro[piperidine-4',1-(1,2,3,4-tetrahydro-beta-carboline)] as a probe defining the extended topographic model of 5-HT1A receptors.

Mokrosz MJ, Duszynska B, Bojarski AJ, Mokrosz JL. Mokrosz MJ, et al. Among authors: bojarski aj. Bioorg Med Chem. 1995 May;3(5):533-8. doi: 10.1016/0968-0896(95)00039-j. Bioorg Med Chem. 1995. PMID: 7648202

3

8-[4-[2-(1,2,3,4-Tetrahydroisoquinolinyl]butyl-8-azaspiro[4.5]decane-7,9-dione: a new 5-HT1A receptor ligand with the same activity profile as buspirone.

Mokrosz JL, Dereń-Wesołek A, Tatarczyńska E, Duszyńska B, Bojarski AJ, Mokrosz MJ, Chojnacka-Wójcik E. Mokrosz JL, et al. Among authors: bojarski aj. J Med Chem. 1996 Mar 1;39(5):1125-9. doi: 10.1021/jm950662c. J Med Chem. 1996. PMID: 8676348

4

On the bioactive conformation of NAN-190 (1) and MP3022 (2), 5-HT(1A) receptor antagonists.

Paluchowska MH, Mokrosz MJ, Bojarski A, Wesołowska A, Borycz J, Charakchieva-Minol S, Chojnacka-Wójcik E. Paluchowska MH, et al. J Med Chem. 1999 Dec 2;42(24):4952-60. doi: 10.1021/jm991045h. J Med Chem. 1999. PMID: 10585205

5

The influence of substitution at aromatic part of 1,2,3,4-tetrahydroisoquinoline on in vitro and in vivo 5-HT(1A)/5-HT(2A) receptor activities of its 1-adamantoyloaminoalkyl derivatives.

Bojarski AJ, Mokrosz MJ, Minol SC, Kozioł A, Wesołowska A, Tatarczyńska E, Kłodzińska A, Chojnacka-Wójcik E. Bojarski AJ, et al. Bioorg Med Chem. 2002 Jan;10(1):87-95. doi: 10.1016/s0968-0896(01)00236-x. Bioorg Med Chem. 2002. PMID: 11738610

6

Active conformation of some arylpiperazine postsynaptic 5-HT(1A) receptor antagonists.

Paluchowska MH, Bojarski AJ, Charakchieva-Minol S, Wesołowska A. Paluchowska MH, et al. Among authors: bojarski aj. Eur J Med Chem. 2002 Apr;37(4):273-83. doi: 10.1016/s0223-5234(01)01312-5. Eur J Med Chem. 2002. PMID: 11960662

7

Substitution mode of the amide fragment in some new N-[omega-[4-(2-methoxyphenyl)piperazin-1-yl]alkyl]pyrid-2(1H)-ones and their 5-HT1A/5-HT2A activity.

Paluchowska MH, Bugno R, Charakchieva-Minol S, Bojarski AJ, Wesołowska A. Paluchowska MH, et al. Among authors: bojarski aj. Pol J Pharmacol. 2001 Jul-Aug;53(4):369-76. Pol J Pharmacol. 2001. PMID: 11990083 Free article.

8

Arylpiperazine derivatives of 3-propyl-beta-tetralonohydantoin as new 5-HT1A and 5-HT2A receptor ligands.

Byrtus H, Pawłowski M, Duszyńska B, Wesołowska A, Chojnacka-Wójcik E, Bojarski AJ. Byrtus H, et al. Among authors: bojarski aj. Pol J Pharmacol. 2001 Jul-Aug;53(4):395-401. Pol J Pharmacol. 2001. PMID: 11990087 Free article.

9

Synthesis and pharmacological evaluation of new arylpiperazines. 3-[4-[4-(3-chlorophenyl)-1-piperazinyl]butyl]-quinazolidin-4-one - a dual serotonin 5-HT(1A)/5-HT(2A) receptor ligand with an anxiolytic-like activity.

Bojarski AJ, Kowalski P, Kowalska T, Duszyńska B, Charakchieva-Minol S, Tatarczyńska E, Kłodzińska A, Chojnacka-Wójcik E. Bojarski AJ, et al. Bioorg Med Chem. 2002 Dec;10(12):3817-27. doi: 10.1016/s0968-0896(02)00349-8. Bioorg Med Chem. 2002. PMID: 12413835

10

Modification of the structure of 4, 6-disubstituted 2-(4-alkyl-1-piperazinyl)pyridines: synthesis and their 5-HT2A receptor activity.

Paluchowska MH, Bojarski AJ, Bugno R, Charakchieva-Minol S, Wesołowska A. Paluchowska MH, et al. Among authors: bojarski aj. Arch Pharm (Weinheim). 2003 Apr;336(2):104-10. doi: 10.1002/ardp.200390006. Arch Pharm (Weinheim). 2003. PMID: 12761763

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