Gay EA - Search Results

1

Indole-Containing Amidinohydrazones as Nonpeptide, Dual RXFP3/4 Agonists: Synthesis, Structure-Activity Relationship, and Molecular Modeling Studies.

Guan D, Rahman MT, Gay EA, Vasukuttan V, Mathews KM, Decker AM, Williams AH, Zhan CG, Jin C. Guan D, et al. Among authors: gay ea. J Med Chem. 2021 Dec 23;64(24):17866-17886. doi: 10.1021/acs.jmedchem.1c01081. Epub 2021 Dec 2. J Med Chem. 2021. PMID: 34855388 Free PMC article.

2

Diarylureas as allosteric modulators of the cannabinoid CB1 receptor: structure-activity relationship studies on 1-(4-chlorophenyl)-3-{3-[6-(pyrrolidin-1-yl)pyridin-2-yl]phenyl}urea (PSNCBAM-1).

German N, Decker AM, Gilmour BP, Gay EA, Wiley JL, Thomas BF, Zhang Y. German N, et al. Among authors: gay ea. J Med Chem. 2014 Sep 25;57(18):7758-69. doi: 10.1021/jm501042u. Epub 2014 Sep 4. J Med Chem. 2014. PMID: 25162172 Free PMC article.

3

Development and validation of a high-throughput calcium mobilization assay for the orphan receptor GPR88.

Decker AM, Gay EA, Mathews KM, Rosa TC, Langston TL, Maitra R, Jin C. Decker AM, et al. Among authors: gay ea. J Biomed Sci. 2017 Mar 27;24(1):23. doi: 10.1186/s12929-017-0330-3. J Biomed Sci. 2017. PMID: 28347302 Free PMC article.

4

Peripherally Selective CB1 Receptor Antagonist Improves Symptoms of Metabolic Syndrome in Mice.

Khan N, Laudermilk L, Ware J, Rosa T, Mathews K, Gay E, Amato G, Maitra R. Khan N, et al. ACS Pharmacol Transl Sci. 2021 Mar 9;4(2):757-764. doi: 10.1021/acsptsci.0c00213. eCollection 2021 Apr 9. ACS Pharmacol Transl Sci. 2021. PMID: 33860199 Free PMC article.

5

Discovery and Characterization of the First Nonpeptide Antagonists for the Relaxin-3/RXFP3 System.

Gay EA, Guan D, Van Voorhies K, Vasukuttan V, Mathews KM, Besheer J, Jin C. Gay EA, et al. J Med Chem. 2022 Jun 9;65(11):7959-7974. doi: 10.1021/acs.jmedchem.2c00508. Epub 2022 May 20. J Med Chem. 2022. PMID: 35594150 Free PMC article.

6

The development of diphenyleneiodonium analogs as GPR3 agonists.

Gay EA, Harris DL, Wilson JW, Blough BE. Gay EA, et al. Bioorg Med Chem Lett. 2023 Oct 1;94:129427. doi: 10.1016/j.bmcl.2023.129427. Epub 2023 Aug 2. Bioorg Med Chem Lett. 2023. PMID: 37541631 Free PMC article.

7

Discovery of 1,3-disubstituted pyrazole peripheral cannabinoid receptor partial agonists.

Amato G, Runyon S, Vasukuttan V, Decker AM, Gay EA, Laudermilk L, Maitra R. Amato G, et al. Among authors: gay ea. Bioorg Med Chem Lett. 2023 Sep 1;93:129430. doi: 10.1016/j.bmcl.2023.129430. Epub 2023 Aug 4. Bioorg Med Chem Lett. 2023. PMID: 37543275 Free PMC article.

8

Novel RXFP3 negative allosteric modulator RLX-33 reduces alcohol self-administration in rats.

Van Voorhies KJ, Liu W, Lovelock DF, Lin S, Liu J, Guan D, Gay EA, Jin C, Besheer J. Van Voorhies KJ, et al. Among authors: gay ea. J Neurochem. 2023 Oct;167(2):204-217. doi: 10.1111/jnc.15949. Epub 2023 Sep 6. J Neurochem. 2023. PMID: 37674350 Free PMC article.

9

Novel Peripherally Selective Cannabinoid Receptor 1 Neutral Antagonist Improves Metabolic Dysfunction-Associated Steatotic Liver Disease in Mice.

Laudermilk LT, Schlosburg JE, Gay EA, Decker AM, Williams A, Runton R, Vasukuttan V, Kotiya A, Amato GS, Maitra R. Laudermilk LT, et al. Among authors: gay ea. ACS Pharmacol Transl Sci. 2024 Aug 8;7(9):2856-2868. doi: 10.1021/acsptsci.4c00356. eCollection 2024 Sep 13. ACS Pharmacol Transl Sci. 2024. PMID: 39296275

10

8,9-dihydroxy-1,2,3,11b-tetrahydrochromeno[4,3,2,-de]isoquinoline (dinoxyline), a high affinity and potent agonist at all dopamine receptor isoforms.

Grubbs RA, Lewis MM, Owens-Vance C, Gay EA, Jassen AK, Mailman RB, Nichols DE. Grubbs RA, et al. Among authors: gay ea. Bioorg Med Chem. 2004 Mar 15;12(6):1403-12. doi: 10.1016/j.bmc.2004.01.008. Bioorg Med Chem. 2004. PMID: 15018913

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