Zappalà M - Search Results

1

Development of novel dipeptide nitriles as inhibitors of rhodesain of Trypanosoma brucei rhodesiense.

Di Chio C, Previti S, Amendola G, Ravichandran R, Wagner A, Cosconati S, Hellmich UA, Schirmeister T, Zappalà M, Ettari R. Di Chio C, et al. Among authors: zappala m. Eur J Med Chem. 2022 Jun 5;236:114328. doi: 10.1016/j.ejmech.2022.114328. Epub 2022 Mar 29. Eur J Med Chem. 2022. PMID: 35385806

2

Discovery of 2,3-diaryl-1,3-thiazolidin-4-ones as potent anti-HIV-1 agents.

Barreca ML, Chimirri A, De Luca L, Monforte AM, Monforte P, Rao A, Zappalà M, Balzarini J, De Clercq E, Pannecouque C, Witvrouw M. Barreca ML, et al. Among authors: zappala m. Bioorg Med Chem Lett. 2001 Jul 9;11(13):1793-6. doi: 10.1016/s0960-894x(01)00304-3. Bioorg Med Chem Lett. 2001. PMID: 11425562

3

Design, synthesis, structure-activity relationships, and molecular modeling studies of 2,3-diaryl-1,3-thiazolidin-4-ones as potent anti-HIV agents.

Barreca ML, Balzarini J, Chimirri A, De Clercq E, De Luca L, Höltje HD, Höltje M, Monforte AM, Monforte P, Pannecouque C, Rao A, Zappalà M. Barreca ML, et al. Among authors: zappala m. J Med Chem. 2002 Nov 21;45(24):5410-3. doi: 10.1021/jm020977+. J Med Chem. 2002. PMID: 12431069

4

Computational strategies in discovering novel non-nucleoside inhibitors of HIV-1 RT.

Barreca ML, Rao A, De Luca L, Zappalà M, Monforte AM, Maga G, Pannecouque C, Balzarini J, De Clercq E, Chimirri A, Monforte P. Barreca ML, et al. Among authors: zappala m. J Med Chem. 2005 May 5;48(9):3433-7. doi: 10.1021/jm049279a. J Med Chem. 2005. PMID: 15857150

5

Pharmacophore-based design of HIV-1 integrase strand-transfer inhibitors.

Barreca ML, Ferro S, Rao A, De Luca L, Zappalà M, Monforte AM, Debyser Z, Witvrouw M, Chimirri A. Barreca ML, et al. Among authors: zappala m. J Med Chem. 2005 Nov 3;48(22):7084-8. doi: 10.1021/jm050549e. J Med Chem. 2005. PMID: 16250669

6

Novel peptidomimetic cysteine protease inhibitors as potential antimalarial agents.

Micale N, Kozikowski AP, Ettari R, Grasso S, Zappalà M, Jeong JJ, Kumar A, Hanspal M, Chishti AH. Micale N, et al. Among authors: zappala m. J Med Chem. 2006 Jun 1;49(11):3064-7. doi: 10.1021/jm060405f. J Med Chem. 2006. PMID: 16722625

7

Development of peptidomimetics with a vinyl sulfone warhead as irreversible falcipain-2 inhibitors.

Ettari R, Nizi E, Di Francesco ME, Dude MA, Pradel G, Vicík R, Schirmeister T, Micale N, Grasso S, Zappalà M. Ettari R, et al. Among authors: zappala m. J Med Chem. 2008 Feb 28;51(4):988-96. doi: 10.1021/jm701141u. Epub 2008 Jan 31. J Med Chem. 2008. PMID: 18232656

8

Nonpeptidic vinyl and allyl phosphonates as falcipain-2 inhibitors.

Ettari R, Nizi E, Di Francesco ME, Micale N, Grasso S, Zappalà M, Vicík R, Schirmeister T. Ettari R, et al. Among authors: zappala m. ChemMedChem. 2008 Jul;3(7):1030-3. doi: 10.1002/cmdc.200800050. ChemMedChem. 2008. PMID: 18428116 No abstract available.

9

Novel peptidomimetics containing a vinyl ester moiety as highly potent and selective falcipain-2 inhibitors.

Ettari R, Micale N, Schirmeister T, Gelhaus C, Leippe M, Nizi E, Di Francesco ME, Grasso S, Zappalà M. Ettari R, et al. Among authors: zappala m. J Med Chem. 2009 Apr 9;52(7):2157-60. doi: 10.1021/jm900047j. J Med Chem. 2009. PMID: 19296600

10

Falcipain-2 inhibitors.

Ettari R, Bova F, Zappalà M, Grasso S, Micale N. Ettari R, et al. Among authors: zappala m. Med Res Rev. 2010 Jan;30(1):136-67. doi: 10.1002/med.20163. Med Res Rev. 2010. PMID: 19526594 Review.

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