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Overcoming undesirable hERG affinity by incorporating fluorine atoms: A case of MAO-B inhibitors derived from 1 H-pyrrolo-[3,2-c]quinolines.
Grychowska K, Olejarz-Maciej A, Blicharz K, Pietruś W, Karcz T, Kurczab R, Koczurkiewicz P, Doroz-Płonka A, Latacz G, Keeri AR, Piska K, Satała G, Pęgiel J, Trybała W, Jastrzębska-Więsek M, Bojarski AJ, Lamaty F, Partyka A, Walczak M, Krawczyk M, Malikowska-Racia N, Popik P, Zajdel P. Grychowska K, et al. Among authors: kurczab r. Eur J Med Chem. 2022 Jun 5;236:114329. doi: 10.1016/j.ejmech.2022.114329. Epub 2022 Mar 29. Eur J Med Chem. 2022. PMID: 35397400 Free article.
The multiobjective based design, synthesis and evaluation of the arylsulfonamide/amide derivatives of aryloxyethyl- and arylthioethyl- piperidines and pyrrolidines as a novel class of potent 5-HT₇ receptor antagonists.
Zajdel P, Kurczab R, Grychowska K, Satała G, Pawłowski M, Bojarski AJ. Zajdel P, et al. Among authors: kurczab r. Eur J Med Chem. 2012 Oct;56:348-60. doi: 10.1016/j.ejmech.2012.07.043. Epub 2012 Aug 4. Eur J Med Chem. 2012. PMID: 22926225
Solid-supported synthesis, molecular modeling, and biological activity of long-chain arylpiperazine derivatives with cyclic amino acid amide fragments as 5-HT(7) and 5-HT(1A) receptor ligands.
Canale V, Guzik P, Kurczab R, Verdie P, Satała G, Kubica B, Pawłowski M, Martinez J, Subra G, Bojarski AJ, Zajdel P. Canale V, et al. Among authors: kurczab r. Eur J Med Chem. 2014 May 6;78:10-22. doi: 10.1016/j.ejmech.2014.03.005. Epub 2014 Mar 5. Eur J Med Chem. 2014. PMID: 24675176
Structure-activity relationships and molecular modeling studies of novel arylpiperazinylalkyl 2-benzoxazolones and 2-benzothiazolones as 5-HT(7) and 5-HT(1A) receptor ligands.
Salerno L, Pittalà V, Modica MN, Siracusa MA, Intagliata S, Cagnotto A, Salmona M, Kurczab R, Bojarski AJ, Romeo G. Salerno L, et al. Among authors: kurczab r. Eur J Med Chem. 2014 Oct 6;85:716-26. doi: 10.1016/j.ejmech.2014.08.023. Epub 2014 Aug 7. Eur J Med Chem. 2014. PMID: 25128671
Towards novel 5-HT7versus 5-HT1A receptor ligands among LCAPs with cyclic amino acid amide fragments: design, synthesis, and antidepressant properties. Part II.
Canale V, Kurczab R, Partyka A, Satała G, Witek J, Jastrzębska-Więsek M, Pawłowski M, Bojarski AJ, Wesołowska A, Zajdel P. Canale V, et al. Among authors: kurczab r. Eur J Med Chem. 2015 Mar 6;92:202-11. doi: 10.1016/j.ejmech.2014.12.041. Epub 2014 Dec 24. Eur J Med Chem. 2015. PMID: 25555143
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