Stoddart LA - Search Results

1

Optimization of Peptide Linker-Based Fluorescent Ligands for the Histamine H₁ Receptor.

Kok ZY, Stoddart LA, Mistry SJ, Mocking TAM, Vischer HF, Leurs R, Hill SJ, Mistry SN, Kellam B. Kok ZY, et al. Among authors: stoddart la. J Med Chem. 2022 Jun 23;65(12):8258-8288. doi: 10.1021/acs.jmedchem.2c00125. Epub 2022 Jun 3. J Med Chem. 2022. PMID: 35734860 Free PMC article.

2

Allosteric interactions across native adenosine-A3 receptor homodimers: quantification using single-cell ligand-binding kinetics.

May LT, Bridge LJ, Stoddart LA, Briddon SJ, Hill SJ. May LT, et al. Among authors: stoddart la. FASEB J. 2011 Oct;25(10):3465-76. doi: 10.1096/fj.11-186296. Epub 2011 Jun 29. FASEB J. 2011. PMID: 21715680 Free PMC article.

3

Highly potent and selective fluorescent antagonists of the human adenosine A₃ receptor based on the 1,2,4-triazolo[4,3-a]quinoxalin-1-one scaffold.

Vernall AJ, Stoddart LA, Briddon SJ, Hill SJ, Kellam B. Vernall AJ, et al. Among authors: stoddart la. J Med Chem. 2012 Feb 23;55(4):1771-82. doi: 10.1021/jm201722y. Epub 2012 Feb 13. J Med Chem. 2012. PMID: 22277057

4

Fragment screening at adenosine-A(3) receptors in living cells using a fluorescence-based binding assay.

Stoddart LA, Vernall AJ, Denman JL, Briddon SJ, Kellam B, Hill SJ. Stoddart LA, et al. Chem Biol. 2012 Sep 21;19(9):1105-15. doi: 10.1016/j.chembiol.2012.07.014. Chem Biol. 2012. PMID: 22999879 Free PMC article.

5

Conversion of a non-selective adenosine receptor antagonist into A3-selective high affinity fluorescent probes using peptide-based linkers.

Vernall AJ, Stoddart LA, Briddon SJ, Ng HW, Laughton CA, Doughty SW, Hill SJ, Kellam B. Vernall AJ, et al. Among authors: stoddart la. Org Biomol Chem. 2013 Sep 14;11(34):5673-82. doi: 10.1039/c3ob41221k. Org Biomol Chem. 2013. PMID: 23881285

6

Fluorescent ligands for G protein-coupled receptors: illuminating receptor-ligand interactions for drug discovery.

Stoddart LA, Briddon SJ, Hill SJ. Stoddart LA, et al. Future Med Chem. 2013 Aug;5(12):1367-9. doi: 10.4155/fmc.13.110. Future Med Chem. 2013. PMID: 23919546 No abstract available.

7

Effect of a toggle switch mutation in TM6 of the human adenosine A₃ receptor on Gi protein-dependent signalling and Gi-independent receptor internalization.

Stoddart LA, Kellam B, Briddon SJ, Hill SJ. Stoddart LA, et al. Br J Pharmacol. 2014 Aug;171(16):3827-44. doi: 10.1111/bph.12739. Br J Pharmacol. 2014. PMID: 24750014 Free PMC article.

8

Direct visualisation of internalization of the adenosine A3 receptor and localization with arrestin3 using a fluorescent agonist.

Stoddart LA, Vernall AJ, Briddon SJ, Kellam B, Hill SJ. Stoddart LA, et al. Neuropharmacology. 2015 Nov;98:68-77. doi: 10.1016/j.neuropharm.2015.04.013. Epub 2015 Apr 30. Neuropharmacology. 2015. PMID: 25937210 Free article.

9

Probing the pharmacology of G protein-coupled receptors with fluorescent ligands.

Stoddart LA, Kilpatrick LE, Briddon SJ, Hill SJ. Stoddart LA, et al. Neuropharmacology. 2015 Nov;98:48-57. doi: 10.1016/j.neuropharm.2015.04.033. Epub 2015 May 13. Neuropharmacology. 2015. PMID: 25979488 Free article. Review.

10

Application of BRET to monitor ligand binding to GPCRs.

Stoddart LA, Johnstone EKM, Wheal AJ, Goulding J, Robers MB, Machleidt T, Wood KV, Hill SJ, Pfleger KDG. Stoddart LA, et al. Nat Methods. 2015 Jul;12(7):661-663. doi: 10.1038/nmeth.3398. Epub 2015 Jun 1. Nat Methods. 2015. PMID: 26030448 Free PMC article.

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