Jacobson KA - Search Results

1

Effects of Purinergic Receptor Deletion or Pharmacologic Modulation on Pulmonary Inflammation in Mice.

Whitehead GS, Karcz TP, Tosh DK, Jung YH, Wen Z, Campbell RG, Gopinatth V, Gao ZG, Jacobson KA, Cook DN. Whitehead GS, et al. Among authors: jacobson ka. ACS Pharmacol Transl Sci. 2022 Oct 5;5(10):973-984. doi: 10.1021/acsptsci.2c00128. eCollection 2022 Oct 14. ACS Pharmacol Transl Sci. 2022. PMID: 36268115 Free PMC article.

2

Site-directed mutagenesis studies of human A(2A) adenosine receptors: involvement of glu(13) and his(278) in ligand binding and sodium modulation.

Gao ZG, Jiang Q, Jacobson KA, Ijzerman AP. Gao ZG, et al. Among authors: jacobson ka. Biochem Pharmacol. 2000 Sep 1;60(5):661-8. doi: 10.1016/s0006-2952(00)00357-9. Biochem Pharmacol. 2000. PMID: 10927024 Free PMC article.

3

Constitutive activation of A(3) adenosine receptors by site-directed mutagenesis.

Chen A, Gao ZG, Barak D, Liang BT, Jacobson KA. Chen A, et al. Among authors: jacobson ka. Biochem Biophys Res Commun. 2001 Jun 15;284(3):596-601. doi: 10.1006/bbrc.2001.5027. Biochem Biophys Res Commun. 2001. PMID: 11396942 Free PMC article.

4

Allosteric modulation of A(3) adenosine receptors by a series of 3-(2-pyridinyl)isoquinoline derivatives.

Gao ZG, Van Muijlwijk-Koezen JE, Chen A, Müller CE, Ijzerman AP, Jacobson KA. Gao ZG, et al. Among authors: jacobson ka. Mol Pharmacol. 2001 Nov;60(5):1057-63. Mol Pharmacol. 2001. PMID: 11641434 Free PMC article.

5

Neoceptor concept based on molecular complementarity in GPCRs: a mutant adenosine A(3) receptor with selectively enhanced affinity for amine-modified nucleosides.

Jacobson KA, Gao ZG, Chen A, Barak D, Kim SA, Lee K, Link A, Rompaey PV, van Calenbergh S, Liang BT. Jacobson KA, et al. J Med Chem. 2001 Nov 22;44(24):4125-36. doi: 10.1021/jm010232o. J Med Chem. 2001. PMID: 11708915 Free PMC article.

6

Identification by site-directed mutagenesis of residues involved in ligand recognition and activation of the human A3 adenosine receptor.

Gao ZG, Chen A, Barak D, Kim SK, Müller CE, Jacobson KA. Gao ZG, et al. Among authors: jacobson ka. J Biol Chem. 2002 May 24;277(21):19056-63. doi: 10.1074/jbc.M110960200. Epub 2002 Mar 12. J Biol Chem. 2002. PMID: 11891221 Free PMC article.

7

2-Chloro-N(6)-cyclopentyladenosine, adenosine A(1) receptor agonist, antagonizes the adenosine A(3) receptor.

Gao ZG, Jacobson KA. Gao ZG, et al. Among authors: jacobson ka. Eur J Pharmacol. 2002 May 17;443(1-3):39-42. doi: 10.1016/s0014-2999(02)01552-2. Eur J Pharmacol. 2002. PMID: 12044789 Free PMC article.

8

Selective allosteric enhancement of agonist binding and function at human A3 adenosine receptors by a series of imidazoquinoline derivatives.

Gao ZG, Kim SG, Soltysiak KA, Melman N, IJzerman AP, Jacobson KA. Gao ZG, et al. Among authors: jacobson ka. Mol Pharmacol. 2002 Jul;62(1):81-9. doi: 10.1124/mol.62.1.81. Mol Pharmacol. 2002. PMID: 12065758 Free PMC article.

9

Structural determinants of A(3) adenosine receptor activation: nucleoside ligands at the agonist/antagonist boundary.

Gao ZG, Kim SK, Biadatti T, Chen W, Lee K, Barak D, Kim SG, Johnson CR, Jacobson KA. Gao ZG, et al. Among authors: jacobson ka. J Med Chem. 2002 Sep 26;45(20):4471-84. doi: 10.1021/jm020211+. J Med Chem. 2002. PMID: 12238926 Free PMC article.

10

Differential allosteric modulation by amiloride analogues of agonist and antagonist binding at A(1) and A(3) adenosine receptors.

Gao ZG, Melman N, Erdmann A, Kim SG, Müller CE, IJzerman AP, Jacobson KA. Gao ZG, et al. Among authors: jacobson ka. Biochem Pharmacol. 2003 Feb 15;65(4):525-34. doi: 10.1016/s0006-2952(02)01556-3. Biochem Pharmacol. 2003. PMID: 12566079 Free PMC article.

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