Baud MGJ - Search Results

1

Discovery of Nanomolar-Affinity Pharmacological Chaperones Stabilizing the Oncogenic p53 Mutant Y220C.

Stephenson Clarke JR, Douglas LR, Duriez PJ, Balourdas DI, Joerger AC, Khadiullina R, Bulatov E, Baud MGJ. Stephenson Clarke JR, et al. Among authors: baud mgj. ACS Pharmacol Transl Sci. 2022 Oct 11;5(11):1169-1180. doi: 10.1021/acsptsci.2c00164. eCollection 2022 Nov 11. ACS Pharmacol Transl Sci. 2022. PMID: 36407959 Free PMC article.

2

Exploiting Transient Protein States for the Design of Small-Molecule Stabilizers of Mutant p53.

Joerger AC, Bauer MR, Wilcken R, Baud MGJ, Harbrecht H, Exner TE, Boeckler FM, Spencer J, Fersht AR. Joerger AC, et al. Among authors: baud mgj. Structure. 2015 Dec 1;23(12):2246-2255. doi: 10.1016/j.str.2015.10.016. Structure. 2015. PMID: 26636255 Free PMC article.

3

Harnessing Fluorine-Sulfur Contacts and Multipolar Interactions for the Design of p53 Mutant Y220C Rescue Drugs.

Bauer MR, Jones RN, Baud MG, Wilcken R, Boeckler FM, Fersht AR, Joerger AC, Spencer J. Bauer MR, et al. ACS Chem Biol. 2016 Aug 19;11(8):2265-74. doi: 10.1021/acschembio.6b00315. Epub 2016 Jun 21. ACS Chem Biol. 2016. PMID: 27267810 Free PMC article.

4

Aminobenzothiazole derivatives stabilize the thermolabile p53 cancer mutant Y220C and show anticancer activity in p53-Y220C cell lines.

Baud MGJ, Bauer MR, Verduci L, Dingler FA, Patel KJ, Horil Roy D, Joerger AC, Fersht AR. Baud MGJ, et al. Eur J Med Chem. 2018 May 25;152:101-114. doi: 10.1016/j.ejmech.2018.04.035. Epub 2018 Apr 21. Eur J Med Chem. 2018. PMID: 29702446 Free PMC article.

5

Key Players in the Mutant p53 Team: Small Molecules, Gene Editing, Immunotherapy.

Chasov V, Mirgayazova R, Zmievskaya E, Khadiullina R, Valiullina A, Stephenson Clarke J, Rizvanov A, Baud MGJ, Bulatov E. Chasov V, et al. Among authors: baud mgj. Front Oncol. 2020 Aug 18;10:1460. doi: 10.3389/fonc.2020.01460. eCollection 2020. Front Oncol. 2020. PMID: 32974171 Free PMC article. Review.

6

Toward Photopharmacological Antimicrobial Chemotherapy Using Photoswitchable Amidohydrolase Inhibitors.

Weston CE, Krämer A, Colin F, Yildiz Ö, Baud MG, Meyer-Almes FJ, Fuchter MJ. Weston CE, et al. ACS Infect Dis. 2017 Feb 10;3(2):152-161. doi: 10.1021/acsinfecdis.6b00148. Epub 2016 Oct 31. ACS Infect Dis. 2017. PMID: 27756124 Free article.

7

Biophysical Survey of Small-Molecule β-Catenin Inhibitors: A Cautionary Tale.

McCoy MA, Spicer D, Wells N, Hoogewijs K, Fiedler M, Baud MGJ. McCoy MA, et al. Among authors: baud mgj. J Med Chem. 2022 May 26;65(10):7246-7261. doi: 10.1021/acs.jmedchem.2c00228. Epub 2022 May 17. J Med Chem. 2022. PMID: 35581674 Free PMC article. Review.

8

Exploring 2-Sulfonylpyrimidine Warheads as Acrylamide Surrogates for Targeted Covalent Inhibition: A BTK Story.

Moraru R, Valle-Argos B, Minton A, Buermann L, Pan S, Wales TE, Joseph RE, Andreotti AH, Strefford JC, Packham G, Baud MGJ. Moraru R, et al. Among authors: baud mgj. J Med Chem. 2024 Aug 22;67(16):13572-13593. doi: 10.1021/acs.jmedchem.3c01927. Epub 2024 Aug 9. J Med Chem. 2024. PMID: 39119945 Free PMC article.

9

Current strategies for the design of PROTAC linkers: a critical review.

Troup RI, Fallan C, Baud MGJ. Troup RI, et al. Among authors: baud mgj. Explor Target Antitumor Ther. 2020;1(5):273-312. doi: 10.37349/etat.2020.00018. Epub 2020 Oct 30. Explor Target Antitumor Ther. 2020. PMID: 36046485 Free PMC article. Review.

10

Is NMR Fragment Screening Fine-Tuned to Assess Druggability of Protein-Protein Interactions?

Dias DM, Van Molle I, Baud MG, Galdeano C, Geraldes CF, Ciulli A. Dias DM, et al. ACS Med Chem Lett. 2014 Jan 9;5(1):23-28. doi: 10.1021/ml400296c. Epub 2013 Nov 3. ACS Med Chem Lett. 2014. PMID: 24436777 Free PMC article.

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