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Conjugation of a 5-nitrofuran-2-oyl moiety to aminoalkylimidazoles produces non-toxic nitrofurans that are efficacious in vitro and in vivo against multidrug-resistant Mycobacterium tuberculosis.
Krasavin M, Lukin A, Vedekhina T, Manicheva O, Dogonadze M, Vinogradova T, Zabolotnykh N, Rogacheva E, Kraeva L, Yablonsky P. Krasavin M, et al. Eur J Med Chem. 2018 Sep 5;157:1115-1126. doi: 10.1016/j.ejmech.2018.08.068. Epub 2018 Aug 29. Eur J Med Chem. 2018. PMID: 30179748
Continued exploration of 1,2,4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX isoform that selectively kill cancer cells in hypoxic environment.
Krasavin M, Shetnev A, Sharonova T, Baykov S, Kalinin S, Nocentini A, Sharoyko V, Poli G, Tuccinardi T, Presnukhina S, Tennikova TB, Supuran CT. Krasavin M, et al. Eur J Med Chem. 2019 Feb 15;164:92-105. doi: 10.1016/j.ejmech.2018.12.049. Epub 2018 Dec 21. Eur J Med Chem. 2019. PMID: 30594030
Attachment of a 5-nitrofuroyl moiety to spirocyclic piperidines produces non-toxic nitrofurans that are efficacious in vitro against multidrug-resistant Mycobacterium tuberculosis.
Krasavin M, Lukin A, Vedekhina T, Manicheva O, Dogonadze M, Vinogradova T, Zabolotnykh N, Rogacheva E, Kraeva L, Sharoyko V, Tennikova TB, Dar'in D, Sokolovich E. Krasavin M, et al. Eur J Med Chem. 2019 Mar 15;166:125-135. doi: 10.1016/j.ejmech.2019.01.050. Epub 2019 Jan 23. Eur J Med Chem. 2019. PMID: 30703656
Pyridazinone-substituted benzenesulfonamides display potent inhibition of membrane-bound human carbonic anhydrase IX and promising antiproliferative activity against cancer cell lines.
Krasavin M, Shetnev A, Baykov S, Kalinin S, Nocentini A, Sharoyko V, Poli G, Tuccinardi T, Korsakov M, Tennikova TB, Supuran CT. Krasavin M, et al. Eur J Med Chem. 2019 Apr 15;168:301-314. doi: 10.1016/j.ejmech.2019.02.044. Epub 2019 Feb 15. Eur J Med Chem. 2019. PMID: 30826507
Novel electrophilic amides amenable by the Ugi reaction perturb thioredoxin system via thioredoxin reductase 1 (TrxR1) inhibition: Identification of DVD-445 as a new lead compound for anticancer therapy.
Jovanović M, Zhukovsky D, Podolski-Renić A, Domračeva I, Žalubovskis R, Senćanski M, Glišić S, Sharoyko V, Tennikova T, Dar'in D, Pešić M, Krasavin M. Jovanović M, et al. Among authors: krasavin m. Eur J Med Chem. 2019 Nov 1;181:111580. doi: 10.1016/j.ejmech.2019.111580. Epub 2019 Aug 1. Eur J Med Chem. 2019. PMID: 31400708
From random to rational: A discovery approach to selective subnanomolar inhibitors of human carbonic anhydrase IV based on the Castagnoli-Cushman multicomponent reaction.
Kalinin S, Nocentini A, Kovalenko A, Sharoyko V, Bonardi A, Angeli A, Gratteri P, Tennikova TB, Supuran CT, Krasavin M. Kalinin S, et al. Among authors: krasavin m. Eur J Med Chem. 2019 Nov 15;182:111642. doi: 10.1016/j.ejmech.2019.111642. Epub 2019 Aug 26. Eur J Med Chem. 2019. PMID: 31476557
154 results