Löser R - Search Results

1

Dipeptide-Derived Alkynes as Potent and Selective Irreversible Inhibitors of Cysteine Cathepsins.

Behring L, Ruiz-Gómez G, Trapp C, Morales M, Wodtke R, Köckerling M, Kopka K, Pisabarro MT, Pietzsch J, Löser R. Behring L, et al. Among authors: loser r. J Med Chem. 2023 Mar 23;66(6):3818-3851. doi: 10.1021/acs.jmedchem.2c01360. Epub 2023 Mar 3. J Med Chem. 2023. PMID: 36867428 Free PMC article.

2

Synthesis of neo-peptidoglycans: an unexpected activity of proteases.

Wehofsky N, Löser R, Buchynskyy A, Welzel P, Bordusa F. Wehofsky N, et al. Among authors: loser r. Angew Chem Int Ed Engl. 2002 Aug 2;41(15):2735-8. doi: 10.1002/1521-3773(20020802)41:15<2735::AID-ANIE2735>3.0.CO;2-E. Angew Chem Int Ed Engl. 2002. PMID: 12203469 No abstract available.

3

Microplate assay for quantitative determination of cathepsin activities in viable cells using derivatives of 4-methoxy-beta-naphthylamide.

Rüttger A, Mollenhauer J, Löser R, Gütschow M, Wiederanders B. Rüttger A, et al. Among authors: loser r. Biotechniques. 2006 Oct;41(4):469-73. doi: 10.2144/000112259. Biotechniques. 2006. PMID: 17068963 Free article.

4

Interaction of papain-like cysteine proteases with dipeptide-derived nitriles.

Löser R, Schilling K, Dimmig E, Gütschow M. Löser R, et al. J Med Chem. 2005 Dec 1;48(24):7688-707. doi: 10.1021/jm050686b. J Med Chem. 2005. PMID: 16302809

5

Dipeptide-derived nitriles containing additional electrophilic sites: potentially irreversible inhibitors of cysteine proteases.

Löser R, Gütschow M. Löser R, et al. J Enzyme Inhib Med Chem. 2009 Dec;24(6):1245-52. doi: 10.3109/14756360902797328. J Enzyme Inhib Med Chem. 2009. PMID: 19912058 Free article.

6

Site-selective radiolabeling of peptides by (18)F-fluorobenzoylation with [(18F)]SFB in solution and on solid phase: a comparative study.

Kuchar M, Pretze M, Kniess T, Steinbach J, Pietzsch J, Löser R. Kuchar M, et al. Among authors: loser r. Amino Acids. 2012 Oct;43(4):1431-43. doi: 10.1007/s00726-012-1216-z. Amino Acids. 2012. PMID: 22302364

7

Use of 3-[(18)F]fluoropropanesulfonyl chloride as a prosthetic agent for the radiolabelling of amines: Investigation of precursor molecules, labelling conditions and enzymatic stability of the corresponding sulfonamides.

Löser R, Fischer S, Hiller A, Köckerling M, Funke U, Maisonial A, Brust P, Steinbach J. Löser R, et al. Beilstein J Org Chem. 2013 May 27;9:1002-11. doi: 10.3762/bjoc.9.115. Print 2013. Beilstein J Org Chem. 2013. PMID: 23766817 Free PMC article.

8

Synthesis and radiopharmacological characterisation of a fluorine-18-labelled azadipeptide nitrile as a potential PET tracer for in vivo imaging of cysteine cathepsins.

Löser R, Bergmann R, Frizler M, Mosch B, Dombrowski L, Kuchar M, Steinbach J, Gütschow M, Pietzsch J. Löser R, et al. ChemMedChem. 2013 Aug;8(8):1330-44. doi: 10.1002/cmdc.201300135. Epub 2013 Jun 19. ChemMedChem. 2013. PMID: 23785011

9

Tissue transglutaminase: an emerging target for therapy and imaging.

Pietsch M, Wodtke R, Pietzsch J, Löser R. Pietsch M, et al. Among authors: loser r. Bioorg Med Chem Lett. 2013 Dec 15;23(24):6528-43. doi: 10.1016/j.bmcl.2013.09.060. Bioorg Med Chem Lett. 2013. PMID: 24432384 Free article. Review.

10

Cyclopeptides containing the DEKS motif as conformationally restricted collagen telopeptide analogues: synthesis and conformational analysis.

Wodtke R, Ruiz-Gómez G, Kuchar M, Pisabarro MT, Novotná P, Urbanová M, Steinbach J, Pietzsch J, Löser R. Wodtke R, et al. Among authors: loser r. Org Biomol Chem. 2015 Feb 14;13(6):1878-96. doi: 10.1039/c4ob02348j. Org Biomol Chem. 2015. PMID: 25503999

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