Vecchio EA - Search Results

1

Biased receptor signalling and intracellular trafficking profiles of structurally distinct formylpeptide receptor 2 agonists.

Peng C, Vecchio EA, Nguyen ATN, De Seram M, Tang R, Keov P, Woodman OL, Chen YC, Baell J, May LT, Zhao P, Ritchie RH, Qin CX. Peng C, et al. Among authors: vecchio ea. Br J Pharmacol. 2024 Nov;181(22):4677-4692. doi: 10.1111/bph.17310. Epub 2024 Aug 18. Br J Pharmacol. 2024. PMID: 39154373

2

Formylpeptide receptor 2: Nomenclature, structure, signalling and translational perspectives: IUPHAR review 35.

Qin CX, Norling LV, Vecchio EA, Brennan EP, May LT, Wootten D, Godson C, Perretti M, Ritchie RH. Qin CX, et al. Among authors: vecchio ea. Br J Pharmacol. 2022 Oct;179(19):4617-4639. doi: 10.1111/bph.15919. Epub 2022 Jul 29. Br J Pharmacol. 2022. PMID: 35797341 Free PMC article. Review.

3

Substituted Pyridazin-3(2 H)-ones as Highly Potent and Biased Formyl Peptide Receptor Agonists.

Deora GS, Qin CX, Vecchio EA, Debono AJ, Priebbenow DL, Brady RM, Beveridge J, Teguh SC, Deo M, May LT, Krippner G, Ritchie RH, Baell JB. Deora GS, et al. Among authors: vecchio ea. J Med Chem. 2019 May 23;62(10):5242-5248. doi: 10.1021/acs.jmedchem.8b01912. Epub 2019 May 13. J Med Chem. 2019. PMID: 31038950

4

The adenosine A_2B G protein-coupled receptor: Recent advances and therapeutic implications.

Vecchio EA, White PJ, May LT. Vecchio EA, et al. Pharmacol Ther. 2019 Jun;198:20-33. doi: 10.1016/j.pharmthera.2019.01.003. Epub 2019 Jan 22. Pharmacol Ther. 2019. PMID: 30677476 Review.

5

New paradigms in adenosine receptor pharmacology: allostery, oligomerization and biased agonism.

Vecchio EA, Baltos JA, Nguyen ATN, Christopoulos A, White PJ, May LT. Vecchio EA, et al. Br J Pharmacol. 2018 Nov;175(21):4036-4046. doi: 10.1111/bph.14337. Epub 2018 Jun 21. Br J Pharmacol. 2018. PMID: 29679502 Free PMC article. Review.

6

Targeting Adenosine Receptors for the Treatment of Cardiac Fibrosis.

Vecchio EA, White PJ, May LT. Vecchio EA, et al. Front Pharmacol. 2017 May 5;8:243. doi: 10.3389/fphar.2017.00243. eCollection 2017. Front Pharmacol. 2017. PMID: 28529484 Free PMC article. Review.

7

Capadenoson, a clinically trialed partial adenosine A₁ receptor agonist, can stimulate adenosine A_2B receptor biased agonism.

Baltos JA, Vecchio EA, Harris MA, Qin CX, Ritchie RH, Christopoulos A, White PJ, May LT. Baltos JA, et al. Among authors: vecchio ea. Biochem Pharmacol. 2017 Jul 1;135:79-89. doi: 10.1016/j.bcp.2017.03.014. Epub 2017 Mar 23. Biochem Pharmacol. 2017. PMID: 28344125

8

Structure of the Adenosine A₁ Receptor Reveals the Basis for Subtype Selectivity.

Glukhova A, Thal DM, Nguyen AT, Vecchio EA, Jörg M, Scammells PJ, May LT, Sexton PM, Christopoulos A. Glukhova A, et al. Among authors: vecchio ea. Cell. 2017 Feb 23;168(5):867-877.e13. doi: 10.1016/j.cell.2017.01.042. Cell. 2017. PMID: 28235198 Free article.

9

Novel Irreversible Agonists Acting at the A₁ Adenosine Receptor.

Jörg M, Glukhova A, Abdul-Ridha A, Vecchio EA, Nguyen AT, Sexton PM, White PJ, May LT, Christopoulos A, Scammells PJ. Jörg M, et al. Among authors: vecchio ea. J Med Chem. 2016 Dec 22;59(24):11182-11194. doi: 10.1021/acs.jmedchem.6b01561. Epub 2016 Dec 13. J Med Chem. 2016. PMID: 27958734

10

Role of the Second Extracellular Loop of the Adenosine A1 Receptor on Allosteric Modulator Binding, Signaling, and Cooperativity.

Nguyen AT, Vecchio EA, Thomas T, Nguyen TD, Aurelio L, Scammells PJ, White PJ, Sexton PM, Gregory KJ, May LT, Christopoulos A. Nguyen AT, et al. Among authors: vecchio ea. Mol Pharmacol. 2016 Dec;90(6):715-725. doi: 10.1124/mol.116.105015. Epub 2016 Sep 28. Mol Pharmacol. 2016. PMID: 27683013

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