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104 results

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Page 1
Use of imidazo[1,5-a]quinoline scaffold as the pharmacophore in the design of bivalent ligands of central benzodiazepine receptors.
Paolino M, Saletti M, Venditti J, Castriconi F, Giuliani G, Maramai S, Toti A, Ghelardini C, Matucci R, Villalobos NA, Anzini M, Cappelli A. Paolino M, et al. Among authors: anzini m. Bioorg Med Chem. 2025 Jan 1;117:118006. doi: 10.1016/j.bmc.2024.118006. Epub 2024 Nov 14. Bioorg Med Chem. 2025. PMID: 39577296 Free article.
Synthesis and structure-activity relationship studies in translocator protein ligands based on a pyrazolo[3,4-b]quinoline scaffold.
Cappelli A, Bini G, Valenti S, Giuliani G, Paolino M, Anzini M, Vomero S, Giorgi G, Giordani A, Stasi LP, Makovec F, Ghelardini C, Di Cesare Mannelli L, Concas A, Porcu P, Biggio G. Cappelli A, et al. Among authors: anzini m. J Med Chem. 2011 Oct 27;54(20):7165-75. doi: 10.1021/jm200770f. Epub 2011 Sep 26. J Med Chem. 2011. PMID: 21916402
Synthesis and structure-activity relationship studies in serotonin 5-HT4 receptor ligands based on a benzo[de][2,6]naphthridine scaffold.
Castriconi F, Paolino M, Giuliani G, Anzini M, Campiani G, Mennuni L, Sabatini C, Lanza M, Caselli G, De Rienzo F, Menziani MC, Sbraccia M, Molinari P, Costa T, Cappelli A. Castriconi F, et al. Among authors: anzini m. Eur J Med Chem. 2014 Jul 23;82:36-46. doi: 10.1016/j.ejmech.2014.05.015. Epub 2014 May 5. Eur J Med Chem. 2014. PMID: 24871995
Design, Synthesis, and Biological Evaluation of Imidazo[1,5-a]quinoline as Highly Potent Ligands of Central Benzodiazepine Receptors.
Cappelli A, Anzini M, Castriconi F, Grisci G, Paolino M, Braile C, Valenti S, Giuliani G, Vomero S, Di Capua A, Betti L, Giannaccini G, Lucacchini A, Ghelardini C, Di Cesare Mannelli L, Frosini M, Ricci L, Giorgi G, Mascia MP, Biggio G. Cappelli A, et al. Among authors: anzini m. J Med Chem. 2016 Apr 14;59(7):3353-72. doi: 10.1021/acs.jmedchem.6b00034. Epub 2016 Mar 24. J Med Chem. 2016. PMID: 26982523
Synthesis, biological evaluation and molecular modeling of novel selective COX-2 inhibitors: sulfide, sulfoxide, and sulfone derivatives of 1,5-diarylpyrrol-3-substituted scaffold.
Reale A, Brogi S, Chelini A, Paolino M, Di Capua A, Giuliani G, Cappelli A, Giorgi G, Chemi G, Grillo A, Valoti M, Sautebin L, Rossi A, Pace S, La Motta C, Di Cesare Mannelli L, Lucarini E, Ghelardini C, Anzini M. Reale A, et al. Among authors: anzini m. Bioorg Med Chem. 2019 Oct 1;27(19):115045. doi: 10.1016/j.bmc.2019.115045. Epub 2019 Aug 9. Bioorg Med Chem. 2019. PMID: 31427145
Design, synthesis and biological evaluation of 7-substituted 4-phenyl-6H-imidazo[1,5-a]thieno[3,2-f] [1,4]diazepines as safe anxiolytic agents.
Di Capua A, Reale A, Paolino M, Chemi G, Brogi S, Cappelli A, Giorgi G, Grande F, Di Cesare Mannelli L, Ghelardini C, Matucci R, Garofalo A, Anzini M. Di Capua A, et al. Among authors: anzini m. Eur J Med Chem. 2020 Aug 15;200:112405. doi: 10.1016/j.ejmech.2020.112405. Epub 2020 May 18. Eur J Med Chem. 2020. PMID: 32492595
Novel multitarget directed ligands inspired by riluzole: A serendipitous synthesis of substituted benzo[b][1,4]thiazepines potentially useful as neuroprotective agents.
Maramai S, Saletti M, Paolino M, Giuliani G, Cazzola J, Spaiardi P, Talpo F, Frosini M, Pifferi A, Ballarotto M, Carotti A, Poggialini F, Vagaggini C, Dreassi E, Giorgi G, Dondio G, Cappelli A, Rosario Biella G, Anzini M. Maramai S, et al. Among authors: anzini m. Bioorg Med Chem. 2024 Oct 1;112:117872. doi: 10.1016/j.bmc.2024.117872. Epub 2024 Aug 13. Bioorg Med Chem. 2024. PMID: 39153378
Novel potent 5-HT(3) receptor ligands based on the pyrrolidone structure: synthesis, biological evaluation, and computational rationalization of the ligand-receptor interaction modalities.
Cappelli A, Anzini M, Vomero S, Mennuni L, Makovec F, Doucet E, Hamon M, Menziani MC, De Benedetti PG, Giorgi G, Ghelardini C, Collina S. Cappelli A, et al. Among authors: anzini m. Bioorg Med Chem. 2002 Mar;10(3):779-801. doi: 10.1016/s0968-0896(01)00332-7. Bioorg Med Chem. 2002. PMID: 11814868
104 results