Childress ES - Search Results

1

Discovery of 4-(5-Membered)Heteroarylether-6-methylpicolinamide Negative Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5.

Childress ES, Capstick RA, Crocker KE, Ledyard ML, Bender AM, Maurer MA, Billard NB, Cho HP, Rodriguez AL, Niswender CM, Peng W, Rook JM, Chang S, Blobaum AL, Boutaud O, Thompson Gray A, Jones CK, Conn PJ, Felts AS, Lindsley CW, Temple KJ. Childress ES, et al. ACS Med Chem Lett. 2024 Nov 18;15(12):2210-2219. doi: 10.1021/acsmedchemlett.4c00481. eCollection 2024 Dec 12. ACS Med Chem Lett. 2024. PMID: 39691522 Free PMC article.

2

Corrigendum to "Design, synthesis and biological evaluation of glucose metabolism inhibitors as anticancer agents" [Bioorg. Chem. 151 (2024) 107665].

Cheng Y, Jones JP, Yu TT, Olzomer EM, Su J, Katen A, Black DS, Hart-Smith G, Childress ES, Beretta M, Wilkins MR, Mateos IA, Santos WL, Hoehn KL, Byrne FL, Kumar N. Cheng Y, et al. Among authors: childress es. Bioorg Chem. 2024 Oct;151:107725. doi: 10.1016/j.bioorg.2024.107725. Epub 2024 Aug 19. Bioorg Chem. 2024. PMID: 39164138 No abstract available.

3

Design, synthesis and biological evaluation of glucose metabolism inhibitors as anticancer agents.

Cheng Y, Jones JP, Yu TT, Olzomer EM, Su J, Katen A, Black DS, Hart-Smith G, Childress ES, Wilkins MR, Mateos IA, Santos WL, Hoehn KL, Byrne FL, Kumar N. Cheng Y, et al. Among authors: childress es. Bioorg Chem. 2024 Oct;151:107665. doi: 10.1016/j.bioorg.2024.107665. Epub 2024 Jul 25. Bioorg Chem. 2024. PMID: 39094508 Free article.

4

Spatial asynchrony and cross-scale climate interactions in populations of a coldwater stream fish.

Valentine GP, Lu X, Childress ES, Dolloff CA, Hitt NP, Kulp MA, Letcher BH, Pregler KC, Rash JM, Hooten MB, Kanno Y. Valentine GP, et al. Among authors: childress es. Glob Chang Biol. 2024 Jan;30(1):e17029. doi: 10.1111/gcb.17029. Epub 2023 Nov 21. Glob Chang Biol. 2024. PMID: 37987546

5

Mitochondrial uncoupler SHC517 reverses obesity in mice without affecting food intake.

Chen SY, Beretta M, Alexopoulos SJ, Shah DP, Olzomer EM, Hargett SR, Childress ES, Salamoun JM, Aleksovska I, Roseblade A, Cranfield C, Rawling T, Quinlan KGR, Morris MJ, Tucker SP, Santos WL, Hoehn KL. Chen SY, et al. Among authors: childress es. Metabolism. 2021 Apr;117:154724. doi: 10.1016/j.metabol.2021.154724. Epub 2021 Feb 4. Metabolism. 2021. PMID: 33548253

6

[1,2,5]Oxadiazolo[3,4-b]pyrazine-5,6-diamine Derivatives as Mitochondrial Uncouplers for the Potential Treatment of Nonalcoholic Steatohepatitis.

Childress ES, Salamoun JM, Hargett SR, Alexopoulos SJ, Chen SY, Shah DP, Santiago-Rivera J, Garcia CJ, Dai Y, Tucker SP, Hoehn KL, Santos WL. Childress ES, et al. J Med Chem. 2020 Mar 12;63(5):2511-2526. doi: 10.1021/acs.jmedchem.9b01440. Epub 2020 Feb 17. J Med Chem. 2020. PMID: 32017849 Free PMC article.

7

Evaluation of Synthetic Cytochrome P₄₅₀-Mimetic Metalloporphyrins To Facilitate "Biomimetic" Biotransformation of a Series of mGlu₅ Allosteric Ligands.

Presley CC, Perry CK, Childress ES, Mulder MJ, Luscombe VB, Rodriguez AL, Niswender CM, Conn PJ, Lindsley CW. Presley CC, et al. Among authors: childress es. ACS Omega. 2019 Jul 26;4(7):12782-12789. doi: 10.1021/acsomega.9b02017. eCollection 2019 Jul 31. ACS Omega. 2019. PMID: 31460402 Free PMC article.

8

Total Synthesis of Hinduchelins A-D, Stereochemical Revision of Hinduchelin A, and Biological Evaluation of Natural and Unnatural Analogues.

Childress ES, Garrison AT, Sheldon JR, Skaar EP, Lindsley CW. Childress ES, et al. J Org Chem. 2019 May 17;84(10):6459-6464. doi: 10.1021/acs.joc.9b00391. Epub 2019 May 8. J Org Chem. 2019. PMID: 31039303 Free PMC article.

9

Preparation of 1,5-Dihydropyrazolo[3',4':5,6]pyrano[3,4- b]pyridines via a Microwave-Assisted, Palladium-Catalyzed Regioselective C-H Heteroarylation of Electron-Rich Pyrazoles.

Garrison AT, Childress ES, Davis DC, Lindsley CW. Garrison AT, et al. Among authors: childress es. J Org Chem. 2019 May 3;84(9):5855-5862. doi: 10.1021/acs.joc.9b00144. Epub 2019 Mar 7. J Org Chem. 2019. PMID: 30807155

10

Discovery of Novel Central Nervous System Penetrant Metabotropic Glutamate Receptor Subtype 2 (mGlu₂) Negative Allosteric Modulators (NAMs) Based on Functionalized Pyrazolo[1,5- a]pyrimidine-5-carboxamide and Thieno[3,2- b]pyridine-5-carboxamide Cores.

Childress ES, Wieting JM, Felts AS, Breiner MM, Long MF, Luscombe VB, Rodriguez AL, Cho HP, Blobaum AL, Niswender CM, Emmitte KA, Conn PJ, Lindsley CW. Childress ES, et al. J Med Chem. 2019 Jan 10;62(1):378-384. doi: 10.1021/acs.jmedchem.8b01266. Epub 2018 Oct 31. J Med Chem. 2019. PMID: 30350962

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