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Off-Target Inhibition of Human Dihydroorotate Dehydrogenase (hDHODH) Highlights Challenges in the Development of Fat Mass and Obesity-Associated Protein (FTO) Inhibitors.
Tarullo M, Fernandez Rodriguez G, Iaiza A, Venezia S, Macone A, Incocciati A, Masciarelli S, Marchioni M, Giorgis M, Lolli ML, Fornaseri F, Proietti L, Grebien F, Rosignoli S, Paiardini A, Rotili D, Mai A, Bochenkova E, Caflisch A, Fazi F, Fatica A. Tarullo M, et al. Among authors: caflisch a. ACS Pharmacol Transl Sci. 2024 Nov 26;7(12):4096-4111. doi: 10.1021/acsptsci.4c00533. eCollection 2024 Dec 13. ACS Pharmacol Transl Sci. 2024. PMID: 39698280
Structure-Based Design of a Potent and Selective YTHDC1 Ligand.
Zálešák F, Nai F, Herok M, Bochenkova E, Bedi RK, Li Y, Errani F, Caflisch A. Zálešák F, et al. Among authors: caflisch a. J Med Chem. 2024 Jun 13;67(11):9516-9535. doi: 10.1021/acs.jmedchem.4c00599. Epub 2024 May 24. J Med Chem. 2024. PMID: 38787793 Free PMC article.
METTL3 Inhibitors for Epitranscriptomic Modulation of Cellular Processes.
Moroz-Omori EV, Huang D, Kumar Bedi R, Cheriyamkunnel SJ, Bochenkova E, Dolbois A, Rzeczkowski MD, Li Y, Wiedmer L, Caflisch A. Moroz-Omori EV, et al. Among authors: caflisch a. ChemMedChem. 2021 Oct 6;16(19):3035-3043. doi: 10.1002/cmdc.202100291. Epub 2021 Jul 29. ChemMedChem. 2021. PMID: 34237194 Free PMC article.
Proteolysis Targeting Chimera Degraders of the METTL3-14 m6A-RNA Methyltransferase.
Errani F, Invernizzi A, Herok M, Bochenkova E, Stamm F, Corbeski I, Romanucci V, Di Fabio G, Zálešák F, Caflisch A. Errani F, et al. Among authors: caflisch a. JACS Au. 2024 Feb 12;4(2):713-729. doi: 10.1021/jacsau.4c00040. eCollection 2024 Feb 26. JACS Au. 2024. PMID: 38425900 Free PMC article.
A Small-Molecule Inhibitor of Lin28.
Roos M, Pradère U, Ngondo RP, Behera A, Allegrini S, Civenni G, Zagalak JA, Marchand JR, Menzi M, Towbin H, Scheuermann J, Neri D, Caflisch A, Catapano CV, Ciaudo C, Hall J. Roos M, et al. Among authors: caflisch a. ACS Chem Biol. 2016 Oct 21;11(10):2773-2781. doi: 10.1021/acschembio.6b00232. Epub 2016 Aug 22. ACS Chem Biol. 2016. PMID: 27548809
278 results