Structure-guided design of potent and selective pyrimidylpyrrole inhibitors of extracellular signal-regulated kinase (ERK) using conformational control.
Aronov AM, Tang Q, Martinez-Botella G, Bemis GW, Cao J, Chen G, Ewing NP, Ford PJ, Germann UA, Green J, Hale MR, Jacobs M, Janetka JW, Maltais F, Markland W, Namchuk MN, Nanthakumar S, Poondru S, Straub J, ter Haar E, Xie X.
Aronov AM, et al. Among authors: markland w.
J Med Chem. 2009 Oct 22;52(20):6362-8. doi: 10.1021/jm900630q.
J Med Chem. 2009.
PMID: 19827834