Stevenson GI - Search Results

1

4,4-Disubstituted piperidine high-affinity NK1 antagonists: structure-activity relationships and in vivo activity.

Stevenson GI, Huscroft I, MacLeod AM, Swain CJ, Cascieri MA, Chicchi GG, Graham MI, Harrison T, Kelleher FJ, Kurtz M, Ladduwahetty T, Merchant KJ, Metzger JM, MacIntyre DE, Sadowski S, Sohal B, Owens AP. Stevenson GI, et al. J Med Chem. 1998 Nov 5;41(23):4623-35. doi: 10.1021/jm980376b. J Med Chem. 1998. PMID: 9804702

2

Novel 5-HT3 antagonists: indol-3-ylspiro(azabicycloalkane-3,5'(4'H)-oxazoles).

Swain CJ, Baker R, Kneen C, Herbert R, Moseley J, Saunders J, Seward EM, Stevenson GI, Beer M, Stanton J, et al. Swain CJ, et al. Among authors: stevenson gi. J Med Chem. 1992 Mar 20;35(6):1019-31. doi: 10.1021/jm00084a007. J Med Chem. 1992. PMID: 1552497

3

4,4-Disubstituted piperidines: a new class of NK1 antagonist.

Stevenson GI, MacLeod AM, Huscroft I, Cascieri MA, Sadowski S, Baker R. Stevenson GI, et al. J Med Chem. 1995 Apr 14;38(8):1264-6. doi: 10.1021/jm00008a003. J Med Chem. 1995. PMID: 7731011 No abstract available.

4

Serine derived NK1 antagonists. 1: The effect of modifications to the serine substituents.

Elliott JM, Cascieri MA, Chicchi G, Davies S, Kelleher FJ, Kurtz M, Ladduwahetty T, Lewis RT, MacLeod AM, Merchant KJ, Sadowski S, Stevenson GI. Elliott JM, et al. Among authors: stevenson gi. Bioorg Med Chem Lett. 1998 Jul 21;8(14):1845-50. doi: 10.1016/s0960-894x(98)00320-5. Bioorg Med Chem Lett. 1998. PMID: 9873445

5

Serine derived NK1 antagonists. 2: A pharmacophore model for arylsulfonamide binding.

Elliott JM, Broughton H, Cascieri MA, Chicchi G, Huscroft IT, Kurtz M, MacLeod AM, Sadowski S, Stevenson GI. Elliott JM, et al. Among authors: stevenson gi. Bioorg Med Chem Lett. 1998 Jul 21;8(14):1851-6. doi: 10.1016/s0960-894x(98)00319-9. Bioorg Med Chem Lett. 1998. PMID: 9873446

6

An efficient protocol for the preparation of primary alcohols bearing a beta-chiral center via an oxazolidinone auxiliary mediated resolution, and application to the synthesis of 4,4-disubstituted piperidine substance P antagonists.

Lewis RT, Ladduwahetty T, Merchant KJ, Keown LE, Hitzel L, Verrier H, Stevenson GI, MacLeod AM. Lewis RT, et al. Among authors: stevenson gi. J Org Chem. 2000 Apr 21;65(8):2615-8. doi: 10.1021/jo9918246. J Org Chem. 2000. PMID: 10789488 No abstract available.

7

Novel 5-HT3 antagonists. Indole oxadiazoles.

Swain CJ, Baker R, Kneen C, Moseley J, Saunders J, Seward EM, Stevenson G, Beer M, Stanton J, Watling K. Swain CJ, et al. J Med Chem. 1991 Jan;34(1):140-51. doi: 10.1021/jm00105a021. J Med Chem. 1991. PMID: 1992112

8

Identification of L-tryptophan derivatives with potent and selective antagonist activity at the NK1 receptor.

MacLeod AM, Merchant KJ, Brookfield F, Kelleher F, Stevenson G, Owens AP, Swain CJ, Casiceri MA, Sadowski S, Ber E, et al. MacLeod AM, et al. J Med Chem. 1994 Apr 29;37(9):1269-74. doi: 10.1021/jm00035a006. J Med Chem. 1994. PMID: 7513763

9

2-Aryl tryptamines: selective high-affinity antagonists for the h5-HT2A receptor.

Stevenson GI, Smith AL, Lewis S, Michie SG, Neduvelil JG, Patel S, Marwood R, Patel S, Castro JL. Stevenson GI, et al. Bioorg Med Chem Lett. 2000 Dec 18;10(24):2697-9. doi: 10.1016/s0960-894x(00)00557-6. Bioorg Med Chem Lett. 2000. PMID: 11133071

10

Purification of the 5-hydroxytryptamine 5-HT3 receptor from NCB20 cells.

McKernan RM, Gillard NP, Quirk K, Kneen CO, Stevenson GI, Swain CJ, Ragan CI. McKernan RM, et al. Among authors: stevenson gi. J Biol Chem. 1990 Aug 15;265(23):13572-7. J Biol Chem. 1990. PMID: 2380174 Free article.

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