Ganellin CR - Search Results

1

Neurochemical and behavioral effects of ciproxifan, a potent histamine H3-receptor antagonist.

Ligneau X, Lin J, Vanni-Mercier G, Jouvet M, Muir JL, Ganellin CR, Stark H, Elz S, Schunack W, Schwartz J. Ligneau X, et al. Among authors: ganellin cr. J Pharmacol Exp Ther. 1998 Nov;287(2):658-66. J Pharmacol Exp Ther. 1998. PMID: 9808693

2

Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain.

Ligneau X, Morisset S, Tardivel-Lacombe J, Gbahou F, Ganellin CR, Stark H, Schunack W, Schwartz JC, Arrang JM. Ligneau X, et al. Among authors: ganellin cr. Br J Pharmacol. 2000 Dec;131(7):1247-50. doi: 10.1038/sj.bjp.0703712. Br J Pharmacol. 2000. PMID: 11090094 Free PMC article.

3

High constitutive activity of native H3 receptors regulates histamine neurons in brain.

Morisset S, Rouleau A, Ligneau X, Gbahou F, Tardivel-Lacombe J, Stark H, Schunack W, Ganellin CR, Schwartz JC, Arrang JM. Morisset S, et al. Among authors: ganellin cr. Nature. 2000 Dec 14;408(6814):860-4. doi: 10.1038/35048583. Nature. 2000. PMID: 11130725

4

Therapeutic implications of constitutive activity of receptors: the example of the histamine H3 receptor.

Schwartz JC, Morisset S, Rouleau A, Ligneau X, Gbahou F, Tardivel-Lacombe J, Stark H, Schunack W, Ganellin CR, Arrang JM. Schwartz JC, et al. Among authors: ganellin cr. J Neural Transm Suppl. 2003;(64):1-16. doi: 10.1007/978-3-7091-6020-6_1. J Neural Transm Suppl. 2003. PMID: 12830926 Review.

5

BF2.649 [1-{3-[3-(4-Chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a nonimidazole inverse agonist/antagonist at the human histamine H3 receptor: Preclinical pharmacology.

Ligneau X, Perrin D, Landais L, Camelin JC, Calmels TP, Berrebi-Bertrand I, Lecomte JM, Parmentier R, Anaclet C, Lin JS, Bertaina-Anglade V, la Rochelle CD, d'Aniello F, Rouleau A, Gbahou F, Arrang JM, Ganellin CR, Stark H, Schunack W, Schwartz JC. Ligneau X, et al. Among authors: ganellin cr. J Pharmacol Exp Ther. 2007 Jan;320(1):365-75. doi: 10.1124/jpet.106.111039. Epub 2006 Sep 27. J Pharmacol Exp Ther. 2007. PMID: 17005916

6

S-[2-(4-imidazolyl)ethyl]isothiourea, a highly specific and potent histamine H3 receptor agonist.

Garbarg M, Arrang JM, Rouleau A, Ligneau X, Tuong MD, Schwartz JC, Ganellin CR. Garbarg M, et al. Among authors: ganellin cr. J Pharmacol Exp Ther. 1992 Oct;263(1):304-10. J Pharmacol Exp Ther. 1992. PMID: 1383495

7

Progress in the proxifan class: heterocyclic congeners as novel potent and selective histamine H(3)-receptor antagonists.

Grassmann S, Sadek B, Ligneau X, Elz S, Ganellin CR, Arrang JM, Schwartz JC, Stark H, Schunack W. Grassmann S, et al. Among authors: ganellin cr. Eur J Pharm Sci. 2002 May;15(4):367-78. doi: 10.1016/s0928-0987(02)00024-6. Eur J Pharm Sci. 2002. PMID: 11988398

8

Piperidino-hydrocarbon compounds as novel non-imidazole histamine H(3)-receptor antagonists.

Meier G, Ligneau X, Pertz HH, Ganellin CR, Schwartz JC, Schunack W, Stark H. Meier G, et al. Among authors: ganellin cr. Bioorg Med Chem. 2002 Aug;10(8):2535-42. doi: 10.1016/s0968-0896(02)00115-3. Bioorg Med Chem. 2002. PMID: 12057642

9

Influence of bulky substituents on histamine h(3) receptor agonist/antagonist properties.

Sasse A, Ligneau X, Rouleau A, Elz S, Ganellin CR, Arrang JM, Schwartz JC, Schunack W, Stark H. Sasse A, et al. Among authors: ganellin cr. J Med Chem. 2002 Aug 29;45(18):4000-10. doi: 10.1021/jm020910m. J Med Chem. 2002. PMID: 12190321

10

Novel nonimidazole histamine H3 receptor antagonists: 1-(4-(phenoxymethyl)benzyl)piperidines and related compounds.

Mikó T, Ligneau X, Pertz HH, Ganellin CR, Arrang JM, Schwartz JC, Schunack W, Stark H. Mikó T, et al. Among authors: ganellin cr. J Med Chem. 2003 Apr 10;46(8):1523-30. doi: 10.1021/jm021084k. J Med Chem. 2003. PMID: 12672253

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

134 results

Search Page

Filters