Garber S - Search Results

1

Design and selection of DMP 850 and DMP 851: the next generation of cyclic urea HIV protease inhibitors.

Rodgers JD, Lam PY, Johnson BL, Wang H, Li R, Ru Y, Ko SS, Seitz SP, Trainor GL, Anderson PS, Klabe RM, Bacheler LT, Cordova B, Garber S, Reid C, Wright MR, Chang CH, Erickson-Viitanen S. Rodgers JD, et al. Among authors: garber s. Chem Biol. 1998 Oct;5(10):597-608. doi: 10.1016/s1074-5521(98)90117-x. Chem Biol. 1998. PMID: 9818151

2

Synthesis, antiviral activity and pharmacokinetics of P1/P1' substituted 3-aminoindazole cyclic urea HIV protease inhibitors.

Kaltenbach RF 3rd, Patel M, Waltermire RE, Harris GD, Stone BR, Klabe RM, Garber S, Bacheler LT, Cordova BC, Logue K, Wright MR, Erickson-Viitanen S, Trainor GL. Kaltenbach RF 3rd, et al. Among authors: garber s. Bioorg Med Chem Lett. 2003 Feb 24;13(4):605-8. doi: 10.1016/s0960-894x(02)01064-8. Bioorg Med Chem Lett. 2003. PMID: 12639540

3

Drug design with a new transition state analog of the hydrated carbonyl: silicon-based inhibitors of the HIV protease.

Chen CA, Sieburth SM, Glekas A, Hewitt GW, Trainor GL, Erickson-Viitanen S, Garber SS, Cordova B, Jeffry S, Klabe RM. Chen CA, et al. Among authors: garber ss. Chem Biol. 2001 Dec;8(12):1161-6. doi: 10.1016/s1074-5521(01)00079-5. Chem Biol. 2001. PMID: 11755395

4

Cyclic urea amides: HIV-1 protease inhibitors with low nanomolar potency against both wild type and protease inhibitor resistant mutants of HIV.

Jadhav PK, Ala P, Woerner FJ, Chang CH, Garber SS, Anton ED, Bacheler LT. Jadhav PK, et al. Among authors: garber ss. J Med Chem. 1997 Jan 17;40(2):181-91. doi: 10.1021/jm960586t. J Med Chem. 1997. PMID: 9003516

5

In vitro anti-human immunodeficiency virus (HIV) activity of XM323, a novel HIV protease inhibitor.

Otto MJ, Reid CD, Garber S, Lam PY, Scarnati H, Bacheler LT, Rayner MM, Winslow DL. Otto MJ, et al. Among authors: garber s. Antimicrob Agents Chemother. 1993 Dec;37(12):2606-11. doi: 10.1128/AAC.37.12.2606. Antimicrob Agents Chemother. 1993. PMID: 8109924 Free PMC article.

6

Improved cyclic urea inhibitors of the HIV-1 protease: synthesis, potency, resistance profile, human pharmacokinetics and X-ray crystal structure of DMP 450.

Hodge CN, Aldrich PE, Bacheler LT, Chang CH, Eyermann CJ, Garber S, Grubb M, Jackson DA, Jadhav PK, Korant B, Lam PY, Maurin MB, Meek JL, Otto MJ, Rayner MM, Reid C, Sharpe TR, Shum L, Winslow DL, Erickson-Viitanen S. Hodge CN, et al. Among authors: garber s. Chem Biol. 1996 Apr;3(4):301-14. doi: 10.1016/s1074-5521(96)90110-6. Chem Biol. 1996. PMID: 8807858

7

Improved P1/P1' substituents for cyclic urea based HIV-1 protease inhibitors: synthesis, structure-activity relationship, and X-ray crystal structure analysis.

Nugiel DA, Jacobs K, Cornelius L, Chang CH, Jadhav PK, Holler ER, Klabe RM, Bacheler LT, Cordova B, Garber S, Reid C, Logue KA, Gorey-Feret LJ, Lam GN, Erickson-Viitanen S, Seitz SP. Nugiel DA, et al. Among authors: garber s. J Med Chem. 1997 May 9;40(10):1465-74. doi: 10.1021/jm960839i. J Med Chem. 1997. PMID: 9154969

8

Nonsymmetric P2/P2' cyclic urea HIV protease inhibitors. Structure-activity relationship, bioavailability, and resistance profile of monoindazole-substituted P2 analogues.

De Lucca GV, Kim UT, Liang J, Cordova B, Klabe RM, Garber S, Bacheler LT, Lam GN, Wright MR, Logue KA, Erickson-Viitanen S, Ko SS, Trainor GL. De Lucca GV, et al. Among authors: garber s. J Med Chem. 1998 Jun 18;41(13):2411-23. doi: 10.1021/jm980103g. J Med Chem. 1998. PMID: 9632373

9

Design and selection of DMP 850 and DMP 851: the next generation of cyclic urea HIV protease inhibitors.

Rodgers JD, Lam PY, Johnson BL, Wang H, Ko SS, Seitz SP, Trainor GL, Anderson PS, Klabe RM, Bacheler LT, Cordova B, Garber S, Reid C, Wright MR, Chang CH, Erickson-Viitanen S. Rodgers JD, et al. Among authors: garber s. Chem Biol. 1998 Nov;5(11):R312. doi: 10.1016/s1074-5521(98)90301-5. Chem Biol. 1998. PMID: 9831533 No abstract available.

10

The synthesis of symmetrical and unsymmetrical P1/P1' cyclic ureas as HIV protease inhibitors.

Patel M, Kaltenbach RF 3rd, Nugiel DA, McHugh RJ Jr, Jadhav PK, Bacheler LT, Cordova BC, Klabe RM, Erickson-Viitanen S, Garber S, Reid C, Seitz SP. Patel M, et al. Among authors: garber s. Bioorg Med Chem Lett. 1998 May 5;8(9):1077-82. doi: 10.1016/s0960-894x(98)00175-9. Bioorg Med Chem Lett. 1998. PMID: 9871711

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