R01 CA109025-03/CA/NCI NIH HHS/United States[Grants and Funding] - Search Results

Year	Number of Results
2007	1
2008	6
2009	2
2010	1
2024	0

1

Design of small-molecule peptidic and nonpeptidic Smac mimetics.

Sun H, Nikolovska-Coleska Z, Yang CY, Qian D, Lu J, Qiu S, Bai L, Peng Y, Cai Q, Wang S. Sun H, et al. Acc Chem Res. 2008 Oct;41(10):1264-77. doi: 10.1021/ar8000553. Acc Chem Res. 2008. PMID: 18937395 Free PMC article.

2

Importance of ligand reorganization free energy in protein-ligand binding-affinity prediction.

Yang CY, Sun H, Chen J, Nikolovska-Coleska Z, Wang S. Yang CY, et al. J Am Chem Soc. 2009 Sep 30;131(38):13709-21. doi: 10.1021/ja9039373. J Am Chem Soc. 2009. PMID: 19736924 Free PMC article.

3

Interaction of a cyclic, bivalent smac mimetic with the x-linked inhibitor of apoptosis protein.

Nikolovska-Coleska Z, Meagher JL, Jiang S, Yang CY, Qiu S, Roller PP, Stuckey JA, Wang S. Nikolovska-Coleska Z, et al. Biochemistry. 2008 Sep 16;47(37):9811-24. doi: 10.1021/bi800785y. Epub 2008 Aug 22. Biochemistry. 2008. PMID: 18717598 Free PMC article.

4

Potent, orally bioavailable diazabicyclic small-molecule mimetics of second mitochondria-derived activator of caspases.

Peng Y, Sun H, Nikolovska-Coleska Z, Qiu S, Yang CY, Lu J, Cai Q, Yi H, Kang S, Yang D, Wang S. Peng Y, et al. J Med Chem. 2008 Dec 25;51(24):8158-62. doi: 10.1021/jm801254r. J Med Chem. 2008. PMID: 19049347 Free PMC article.

5

Design, synthesis, and evaluation of potent, nonpeptidic mimetics of second mitochondria-derived activator of caspases.

Sun W, Nikolovska-Coleska Z, Qin D, Sun H, Yang CY, Bai L, Qiu S, Wang Y, Ma D, Wang S. Sun W, et al. J Med Chem. 2009 Feb 12;52(3):593-6. doi: 10.1021/jm801101z. J Med Chem. 2009. PMID: 19138149 Free PMC article.

6

Design, synthesis, and characterization of a potent, nonpeptide, cell-permeable, bivalent Smac mimetic that concurrently targets both the BIR2 and BIR3 domains in XIAP.

Sun H, Nikolovska-Coleska Z, Lu J, Meagher JL, Yang CY, Qiu S, Tomita Y, Ueda Y, Jiang S, Krajewski K, Roller PP, Stuckey JA, Wang S. Sun H, et al. J Am Chem Soc. 2007 Dec 12;129(49):15279-94. doi: 10.1021/ja074725f. Epub 2007 Nov 14. J Am Chem Soc. 2007. PMID: 17999504 Free PMC article.

7

Structure-based design, synthesis, evaluation, and crystallographic studies of conformationally constrained Smac mimetics as inhibitors of the X-linked inhibitor of apoptosis protein (XIAP).

Sun H, Stuckey JA, Nikolovska-Coleska Z, Qin D, Meagher JL, Qiu S, Lu J, Yang CY, Saito NG, Wang S. Sun H, et al. J Med Chem. 2008 Nov 27;51(22):7169-80. doi: 10.1021/jm8006849. J Med Chem. 2008. PMID: 18954041 Free PMC article.

8

Cyclopeptide Smac mimetics as antagonists of IAP proteins.

Sun H, Liu L, Lu J, Qiu S, Yang CY, Yi H, Wang S. Sun H, et al. Bioorg Med Chem Lett. 2010 May 15;20(10):3043-6. doi: 10.1016/j.bmcl.2010.03.114. Bioorg Med Chem Lett. 2010. PMID: 20443226 Free PMC article.

9

SM-164: a novel, bivalent Smac mimetic that induces apoptosis and tumor regression by concurrent removal of the blockade of cIAP-1/2 and XIAP.

Lu J, Bai L, Sun H, Nikolovska-Coleska Z, McEachern D, Qiu S, Miller RS, Yi H, Shangary S, Sun Y, Meagher JL, Stuckey JA, Wang S. Lu J, et al. Cancer Res. 2008 Nov 15;68(22):9384-93. doi: 10.1158/0008-5472.CAN-08-2655. Cancer Res. 2008. PMID: 19010913 Free PMC article.

10

Design, synthesis, and evaluation of tricyclic, conformationally constrained small-molecule mimetics of second mitochondria-derived activator of caspases.

Zhang B, Nikolovska-Coleska Z, Zhang Y, Bai L, Qiu S, Yang CY, Sun H, Wang S, Wu Y. Zhang B, et al. J Med Chem. 2008 Dec 11;51(23):7352-5. doi: 10.1021/jm801146d. J Med Chem. 2008. PMID: 19012392 Free PMC article.

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